Search Ontology:
ChEBI

osimertinib mesylate

Term ID
CHEBI:90948
Synonyms
  • AZD9291 mesylate
  • N-(2-{[2-(dimethylamino)ethyl](methyl)amino}-4-methoxy-5-{[4-(1-methyl-1H-indol-3-yl)pyrimidin-2-yl]amino}phenyl)prop-2-enamide methanesulfonate
  • osimertinib mesilate
  • osimertinib mesylate
  • osimertinib methanesulfonate
  • osimertinib monomesylate
  • Tagrisso
Definition
A methanesulfonate (mesylate) salt prepared from equimolar amounts of osimertinib and methanesulfonic acid. It is used for treatment of EGFR T790M mutation positive non-small cell lung cancer.
References
  • cas:1421373-66-1
  • kegg.drug:D10766
  • pubmed:26515464
  • pubmed:26620497
  • pubmed:26720284
  • pubmed:26720671
  • pubmed:26729184
  • pubmed:27641462
  • pubmed:27660466
  • pubmed:27923840
  • pubmed:28710746
  • pubmed:29180936
  • pubmed:29998228
  • pubmed:30073261
  • pubmed:30643560
  • pubmed:32211870
  • pubmed:33755621
  • pubmed:34156056
  • pubmed:34564820
  • pubmed:34723634
  • reaxys:23334374
Ontology
ChEBI  ( EBI )
Relationships
Phenotype
Phenotype resulting from osimertinib mesylate
Phenotype where environments contain osimertinib mesylate
Phenotype modified by environments containing osimertinib mesylate
Phenotype affecting osimertinib mesylate
Human Disease Model